Cardiff University | Prifysgol Caerdydd ORCA
Online Research @ Cardiff 
WelshClear Cookie - decide language by browser settings

Browse by Current Cardiff authors

Up a level
Export as [feed] Atom [feed] RSS 1.0 [feed] RSS 2.0
Number of items: 18.

Flude, Ben M., Nannetti, Giulio, Mitchell, Paige, Compton, Nina, Richards, Chloe, Heurich, Meike, Brancale, Andrea, Ferla, Salvatore and Bassetto, Marcella 2021. Targeting the complement serine protease MASP-2 as a therapeutic strategy for coronavirus infections. Viruses 13 (2) , 312. 10.3390/v13020312
file

Massari, Serena, Bertagnin, Chiara, Pismataro, Maria Chiara, Donnadio, Anna, Nannetti, Giulio, Felicetti, Tommaso, Di Bona, Stefano, Nizi, Maria Giulia, Tensi, Leonardo, Manfroni, Giuseppe, Loza, Maria Isabel, Sabatini, Stefano, Cecchetti, Violetta, Brea, Jose, Goracci, Laura, Loregian, Arianna and Tabarrini, Oriana 2021. Synthesis and characterization of 1,2,4-triazolo[1,5-a]pyrimidine-2-carboxamide-based compounds targeting the PA-PB1 interface of influenza A virus polymerase. European Journal of Medicinal Chemistry 209 , 112944. 10.1016/j.ejmech.2020.112944
file

Nannetti, Giulio, Massari, Serena, Mercorelli, Beatrice, Bertagnin, Chiara, Desantis, Jenny, Palù, Giorgio, Tabarrini, Oriana and Loregian, Arianna 2019. Potent and broad-spectrum cycloheptathiophene-3-carboxamide compounds that target the PA-PB1 interaction of influenza virus RNA polymerase and possess a high barrier to drug resistance. Antiviral Research 165 , pp. 55-64. 10.1016/j.antiviral.2019.03.003
file

Nannetti, Giulio, Pagni, Silvana, Palù, Giorgio and Loregian, Arianna 2018. A sensitive and validated HPLC-UV method for the quantitative determination of the new antifungal drug isavuconazole in human plasma. Biomedical Chromatography 32 (11) , e4333. 10.1002/bmc.4333
file

D'Agostino, Ilaria, Giacchello, Ilaria, Nannetti, Giulio, Fallacara, Anna Lucia, Deodato, Davide, Musumeci, Francesca, Grossi, Giancarlo, Palù, Giorgio, Cau, Ylenia, Trist, Iuni Margaret, Loregian, Arianna, Schenone, Silvia and Botta, Maurizio 2018. Synthesis and biological evaluation of a library of hybrid derivatives as inhibitors of influenza virus PA-PB1 interaction. European Journal of Medicinal Chemistry 157 , pp. 743-758. 10.1016/j.ejmech.2018.08.032
file

Messa, Lorenzo, Celegato, Marta, Bertagnin, Chiara, Mercorelli, Beatrice, Nannetti, Giulio, Palù, Giorgio and Loregian, Arianna 2018. A quantitative LumiFluo assay to test inhibitory compounds blocking p53 degradation induced by human papillomavirus oncoprotein E6 in living cells. Scientific Reports 8 (1) , 6020. 10.1038/s41598-018-24470-4
file

Desantis, Jenny, Nannetti, Giulio, Massari, Serena, Barreca, Maria Letizia, Manfroni, Giuseppe, Cecchetti, Violetta, Palù, Giorgio, Goracci, Laura, Loregian, Arianna and Tabarrini, Oriana 2017. Exploring the cycloheptathiophene-3-carboxamide scaffold to disrupt the interactions of the influenza polymerase subunits and obtain potent anti-influenza activity. European Journal of Medicinal Chemistry 138 , pp. 128-139. 10.1016/j.ejmech.2017.06.015
file

Massari, Serena, Desantis, Jenny, Nannetti, Giulio, Sabatini, Stefano, Tortorella, Sara, Goracci, Laura, Cecchetti, Violetta, Loregian, Arianna and Tabarrini, Oriana 2017. Efficient and regioselective one-step synthesis of 7-aryl-5-methyl- and 5-aryl-7-methyl-2-amino-[1,2,4]triazolo[1,5-a]pyrimidine derivatives. Organic and Biomolecular Chemistry 15 (37) , pp. 7944-7955. 10.1039/C7OB02085F
file

Nannetti, Giulio, Messa, Lorenzo, Celegato, Marta, Pagni, Silvana, Basso, Monica, Parisi, Saverio G., Palù, Giorgio and Loregian, Arianna 2017. Development and validation of a simple and robust HPLC method with UV detection for quantification of the hepatitis C virus inhibitor daclatasvir in human plasma. Journal of Pharmaceutical and Biomedical Analysis 134 , pp. 275-281. 10.1016/j.jpba.2016.11.032
file

Parisi, Saverio G., Loregian, Arianna, Andreis, Samantha, Nannetti, Giulio, Cavinato, Silvia, Basso, Monica, Scaggiante, Renzo, Dal Bello, Federico, Messa, Lorenzo, Cattelan, Anna Maria and Palù, Giorgio 2016. Daclatasvir plasma level and resistance selection in HIV patients with hepatitis C virus cirrhosis treated with daclatasvir, sofosbuvir, and ribavirin. International Journal of Infectious Diseases 49 , p. 151. 10.1016/j.ijid.2016.06.020
file

Trist, Iuni M. L., Nannetti, Giulio, Tintori, Cristina, Fallacara, Anna Lucia, Deodato, Davide, Mercorelli, Beatrice, Palù, Giorgio, Wijtmans, Maikel, Gospodova, Tzveta, Edink, Ewald, Verheij, Mark, de Esch, Iwan, Viteva, Lilia, Loregian, Arianna and Botta, Maurizio 2016. 4,6-diphenylpyridines as promising novel anti-influenza agents targeting the PA–PB1 protein–protein interaction: structure–activity relationships exploration with the aid of molecular modeling. Journal of Medicinal Chemistry 59 (6) , pp. 2688-2703. 10.1021/acs.jmedchem.5b01935
file

Nannetti, Giulio, Pagni, Silvana, Parisi, Saverio G., Alberti, Alfredo, Loregian, Arianna and Palù, Giorgio 2016. Development of a simple HPLC-UV method for the determination of the hepatitis C virus inhibitor simeprevir in human plasma. Journal of Pharmaceutical and Biomedical Analysis 121 , pp. 197-203. 10.1016/j.jpba.2016.01.019
file

Mercorelli, Beatrice, Luganini, Anna, Nannetti, Giulio, Tabarrini, Oriana, Palù, Giorgio, Gribaudo, Giorgio and Loregian, Arianna 2016. Drug repurposing approach identifies inhibitors of the prototypic viral transcription Factor IE2 that block human cytomegalovirus replication. Cell Chemical Biology 23 (3) , pp. 340-351. 10.1016/j.chembiol.2015.12.012
file

Massari, Serena, Nannetti, Giulio, Desantis, Jenny, Muratore, Giulia, Sabatini, Stefano, Manfroni, Giuseppe, Mercorelli, Beatrice, Cecchetti, Violetta, Palù, Giorgio, Cruciani, Gabriele, Loregian, Arianna, Goracci, Laura and Tabarrini, Oriana 2015. A broad anti-influenza hybrid small molecule that potently disrupts the interaction of polymerase acidic protein-basic protein 1 (PA-PB1) subunits. Journal of Medicinal Chemistry 58 (9) , pp. 3830-3842. 10.1021/acs.jmedchem.5b00012
file

Loregian, Arianna, Mercorelli, Beatrice, Nannetti, Giulio, Compagnin, Chiara and Palù, Giorgio 2014. Antiviral strategies against influenza virus: towards new therapeutic approaches. Cellular and Molecular Life Sciences 71 (19) , pp. 3659-3683. 10.1007/s00018-014-1615-2
file

Lepri, Susan, Nannetti, Giulio, Muratore, Giulia, Cruciani, Gabriele, Ruzziconi, Renzo, Mercorelli, Beatrice, Palù, Giorgio, Loregian, Arianna and Goracci, Laura 2014. Optimization of small-molecule inhibitors of influenza virus polymerase: From thiophene-3-carboxamide to polyamido scaffolds. Journal of Medicinal Chemistry 57 (10) , pp. 4337-4350. 10.1021/jm500300r
file

Massari, Serena, Nannetti, Giulio, Goracci, Laura, Sancineto, Luca, Muratore, Giulia, Sabatini, Stefano, Manfroni, Giuseppe, Mercorelli, Beatrice, Cecchetti, Violetta, Facchini, Marzia, Palù, Giorgio, Cruciani, Gabriele, Loregian, Arianna and Tabarrini, Oriana 2013. Structural investigation of Cycloheptathiophene-3-carboxamide derivatives targeting influenza virus polymerase assembly. Journal of Medicinal Chemistry 56 (24) , pp. 10118-10131. 10.1021/jm401560v
file

Saladini, Francesco, Foley, Brian T., Rosi, Andrea, Vicenti, Ilaria, Nannetti, Giulio, Meini, Genny, Razzolini, Francesca and Zazzi, Maurizio 2012. Near full-length sequence analysis of HIV Type 1 BF recombinants from Italy. AIDS Research and Human Retroviruses 28 (3) , p. 299. 10.1089/aid.2011.0002
file

This list was generated on Thu Jan 6 04:29:57 2022 GMT.