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Up a levelNumber of items: 7.
Gomaa, Mohamed S., Lim, Andrew S. T., Lau, Sze C. W., Watts, Ann-Marie, Illingworth, N. A., Bridgens, C. E., Veal, G. J., Redfern, C. P. F., Brancale, Andrea  ORCID: https://orcid.org/0000-0002-9728-3419, Armstrong, J. L. and Simons, Claire ORCID: https://orcid.org/0000-0002-9487-1100
2012.
Synthesis and CYP26A1 inhibitory activity of novel methyl 3-[4-(arylamino)phenyl]-3-(azole)-2,2-dimethylpropanoates.
Bioorganic & Medicinal Chemistry
20
(20)
, pp. 6080-6088.
10.1016/j.bmc.2012.08.044
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Gomaa, Mohamed S., Bridgens, C. E., Illingworth, N. A., Veal, G. J., Redfern, C. P. F., Brancale, Andrea ORCID: https://orcid.org/0000-0002-9728-3419, Armstrong, J. L. and Simons, Claire ORCID: https://orcid.org/0000-0002-9487-1100
2012.
Novel retinoic acid 4-hydroxylase (CYP26) inhibitors based on a 3-(1H-imidazol- and triazol-1-yl)-2,2-dimethyl-3-(4-(phenylamino)phenyl)propyl scaffold.
Bioorganic & Medicinal Chemistry
20
(14)
, pp. 4201-4207.
10.1016/j.bmc.2012.05.076
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Gomaa, Mohamed Sayed, Bridgens, Caroline E., Veal, Gareth J., Redfern, Christoper P.F., Brancale, Andrea ORCID: https://orcid.org/0000-0002-9728-3419, Armstrong, Jane L. and Simons, Claire ORCID: https://orcid.org/0000-0002-9487-1100
2011.
Synthesis and biological evaluation of 3-(1H-Imidazol- and Triazol-1-yl)-2,2-Dimethyl-3-[4-(Naphthalen-2-ylamino)phenyl]propyl derivatives as small molecule inhibitors of Retinoic Acid 4-Hydroxylase (CYP26).
Journal of Medicinal Chemistry
54
(19)
, pp. 6803-6811.
10.1021/jm200695m
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Gomaa, Mohamed Sayed, Bridgens, Caroline E., Aboraia, Ahmed, Veal, Gareth J., Redfern, Christopher P. F., Brancale, Andrea ORCID: https://orcid.org/0000-0002-9728-3419, Armstrong, Jane L. and Simons, Claire ORCID: https://orcid.org/0000-0002-9487-1100
2011.
Small molecule inhibitors of retinoic acid 4-hydroxylase (CYP26): Synthesis and biological evaluation of imidazole methyl 3-(4-(aryl-2-ylamino)phenyl)propanoates.
Journal of Medicinal Chemistry
54
(8)
, pp. 2778-2791.
10.1021/jm101583w
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Aboraia, Ahmed S., Yee, Sook Wah, Gomaa, Mohamed Sayed, Shah, Nikhil, Robotham, Anna C., Makowski, Bart, Prosser, David, Brancale, Andrea ORCID: https://orcid.org/0000-0002-9728-3419, Jones, Glenville and Simons, Claire ORCID: https://orcid.org/0000-0002-9487-1100
2010.
Synthesis and CYP24A1 inhibitory activity of N-(2-(1H-imidazol-1-yl)-2-phenylethyl)arylamides.
Bioorganic & Medicinal Chemistry
18
(14)
, pp. 4939-4946.
10.1016/j.bmc.2010.06.011
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Gomaa, Mohamed Sayed, Simons, Claire ORCID: https://orcid.org/0000-0002-9487-1100 and Brancale, Andrea ORCID: https://orcid.org/0000-0002-9728-3419
2007.
Homology model of 1α,25-dihydroxyvitamin D3 24-hydroxylase cytochrome P450 24A1 (CYP24A1): Active site architecture and ligand binding.
The Journal of Steroid Biochemistry and Molecular Biology
104
(1-2)
, pp. 53-60.
10.1016/j.jsbmb.2006.09.041
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Yee, Sook Wah, Jarno, Laetitia, Gomaa, Mohamed Sayed, Elford, Carole, Ooi, Liling, Coogan, Michael Peter, McClelland, Richard Andrew, Nicholson, Robert Ian, Evans, Bronwen Alice James ORCID: https://orcid.org/0000-0002-3082-1008, Brancale, Andrea ORCID: https://orcid.org/0000-0002-9728-3419 and Simons, Claire ORCID: https://orcid.org/0000-0002-9487-1100
2005.
Novel tetralone-derived retinoic acid metabolism blocking agents: synthesis and in vitro evaluation with liver microsomal and MCF-7 CYP26A1 cell assays.
Journal of Medicinal Chemistry
48
(23)
, pp. 7123-7131.
10.1021/jm0501681
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