Nannetti, Giulio ORCID: https://orcid.org/0000-0003-3227-1537, Mercorelli, Beatrice, Bazzacco, Alessandro, Santi, Nicolo ORCID: https://orcid.org/0000-0001-6361-5457, Celegato, Marta, Ferla, Salvatore, Sturlese, Mattia, Buurma, Niklaas J. ORCID: https://orcid.org/0000-0003-0260-5057, Brancale, Andrea ORCID: https://orcid.org/0000-0002-9728-3419 and Loregian, Arianna
2025.
New dengue virus inhibitors targeting NS3-NS5 interaction identified by in silico screening.
Frontiers in Microbiology
16
, 1663404.
10.3389/fmicb.2025.1663404
|
|
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Giancotti, Gilda, Nannetti, Giulio ORCID: https://orcid.org/0000-0003-3227-1537, Padalino, Gilda, Landini, Martina, Santos-Ferreira, Nanci, Van Dycke, Jana, Naccarato, Valentina, Patel, Usheer, Silvestri, Romano, Neyts, Johan, Gozalbo-Rovira, Roberto, Rodríguez-Díaz, Jésus, Rocha-Pereira, Joana, Brancale, Andrea ORCID: https://orcid.org/0000-0002-9728-3419, Ferla, Salvatore ORCID: https://orcid.org/0000-0002-5918-9237 and Bassetto, Marcella ORCID: https://orcid.org/0000-0002-2491-5868
2022.
Structural investigations on novel non-nucleoside inhibitors of human norovirus polymerase.
Viruses
15
(1)
, 74.
10.3390/v15010074
|
|
|
Flude, Ben M., Nannetti, Giulio ORCID: https://orcid.org/0000-0003-3227-1537, Mitchell, Paige, Compton, Nina, Richards, Chloe, Heurich, Meike ORCID: https://orcid.org/0000-0003-0105-2702, Brancale, Andrea ORCID: https://orcid.org/0000-0002-9728-3419, Ferla, Salvatore ORCID: https://orcid.org/0000-0002-5918-9237 and Bassetto, Marcella ORCID: https://orcid.org/0000-0002-2491-5868
2021.
Targeting the complement serine protease MASP-2 as a therapeutic strategy for coronavirus infections.
Viruses
13
(2)
, 312.
10.3390/v13020312
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|
|
Massari, Serena, Bertagnin, Chiara, Pismataro, Maria Chiara, Donnadio, Anna, Nannetti, Giulio ORCID: https://orcid.org/0000-0003-3227-1537, Felicetti, Tommaso, Di Bona, Stefano, Nizi, Maria Giulia, Tensi, Leonardo, Manfroni, Giuseppe, Loza, Maria Isabel, Sabatini, Stefano, Cecchetti, Violetta, Brea, Jose, Goracci, Laura, Loregian, Arianna and Tabarrini, Oriana
2021.
Synthesis and characterization of 1,2,4-triazolo[1,5-a]pyrimidine-2-carboxamide-based compounds targeting the PA-PB1 interface of influenza A virus polymerase.
European Journal of Medicinal Chemistry
209
, 112944.
10.1016/j.ejmech.2020.112944
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|
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Nannetti, Giulio ORCID: https://orcid.org/0000-0003-3227-1537, Massari, Serena, Mercorelli, Beatrice, Bertagnin, Chiara, Desantis, Jenny, Palù, Giorgio, Tabarrini, Oriana and Loregian, Arianna
2019.
Potent and broad-spectrum cycloheptathiophene-3-carboxamide compounds that target the PA-PB1 interaction of influenza virus RNA polymerase and possess a high barrier to drug resistance.
Antiviral Research
165
, pp. 55-64.
10.1016/j.antiviral.2019.03.003
|
|
|
Nannetti, Giulio ORCID: https://orcid.org/0000-0003-3227-1537, Pagni, Silvana, Palù, Giorgio and Loregian, Arianna
2018.
A sensitive and validated HPLC-UV method for the quantitative determination of the new antifungal drug isavuconazole in human plasma.
Biomedical Chromatography
32
(11)
, e4333.
10.1002/bmc.4333
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D'Agostino, Ilaria, Giacchello, Ilaria, Nannetti, Giulio ORCID: https://orcid.org/0000-0003-3227-1537, Fallacara, Anna Lucia, Deodato, Davide, Musumeci, Francesca, Grossi, Giancarlo, Palù, Giorgio, Cau, Ylenia, Trist, Iuni Margaret, Loregian, Arianna, Schenone, Silvia and Botta, Maurizio
2018.
Synthesis and biological evaluation of a library of hybrid derivatives as inhibitors of influenza virus PA-PB1 interaction.
European Journal of Medicinal Chemistry
157
, pp. 743-758.
10.1016/j.ejmech.2018.08.032
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Messa, Lorenzo, Celegato, Marta, Bertagnin, Chiara, Mercorelli, Beatrice, Nannetti, Giulio ORCID: https://orcid.org/0000-0003-3227-1537, Palù, Giorgio and Loregian, Arianna
2018.
A quantitative LumiFluo assay to test inhibitory compounds blocking p53 degradation induced by human papillomavirus oncoprotein E6 in living cells.
Scientific Reports
8
(1)
, 6020.
10.1038/s41598-018-24470-4
|
|
|
Desantis, Jenny, Nannetti, Giulio ORCID: https://orcid.org/0000-0003-3227-1537, Massari, Serena, Barreca, Maria Letizia, Manfroni, Giuseppe, Cecchetti, Violetta, Palù, Giorgio, Goracci, Laura, Loregian, Arianna and Tabarrini, Oriana
2017.
Exploring the cycloheptathiophene-3-carboxamide scaffold to disrupt the interactions of the influenza polymerase subunits and obtain potent anti-influenza activity.
European Journal of Medicinal Chemistry
138
, pp. 128-139.
10.1016/j.ejmech.2017.06.015
|
|
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Massari, Serena, Desantis, Jenny, Nannetti, Giulio ORCID: https://orcid.org/0000-0003-3227-1537, Sabatini, Stefano, Tortorella, Sara, Goracci, Laura, Cecchetti, Violetta, Loregian, Arianna and Tabarrini, Oriana
2017.
Efficient and regioselective one-step synthesis of 7-aryl-5-methyl- and 5-aryl-7-methyl-2-amino-[1,2,4]triazolo[1,5-a]pyrimidine derivatives.
Organic and Biomolecular Chemistry
15
(37)
, pp. 7944-7955.
10.1039/C7OB02085F
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|
Nannetti, Giulio ORCID: https://orcid.org/0000-0003-3227-1537, Messa, Lorenzo, Celegato, Marta, Pagni, Silvana, Basso, Monica, Parisi, Saverio G., Palù, Giorgio and Loregian, Arianna
2017.
Development and validation of a simple and robust HPLC method with UV detection for quantification of the hepatitis C virus inhibitor daclatasvir in human plasma.
Journal of Pharmaceutical and Biomedical Analysis
134
, pp. 275-281.
10.1016/j.jpba.2016.11.032
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|
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Parisi, Saverio G., Loregian, Arianna, Andreis, Samantha, Nannetti, Giulio ORCID: https://orcid.org/0000-0003-3227-1537, Cavinato, Silvia, Basso, Monica, Scaggiante, Renzo, Dal Bello, Federico, Messa, Lorenzo, Cattelan, Anna Maria and Palù, Giorgio
2016.
Daclatasvir plasma level and resistance selection in HIV patients with hepatitis C virus cirrhosis treated with daclatasvir, sofosbuvir, and ribavirin.
International Journal of Infectious Diseases
49
, p. 151.
10.1016/j.ijid.2016.06.020
|
|
|
Trist, Iuni M. L., Nannetti, Giulio ORCID: https://orcid.org/0000-0003-3227-1537, Tintori, Cristina, Fallacara, Anna Lucia, Deodato, Davide, Mercorelli, Beatrice, Palù, Giorgio, Wijtmans, Maikel, Gospodova, Tzveta, Edink, Ewald, Verheij, Mark, de Esch, Iwan, Viteva, Lilia, Loregian, Arianna and Botta, Maurizio
2016.
4,6-diphenylpyridines as promising novel anti-influenza agents targeting the PA–PB1 protein–protein interaction: structure–activity relationships exploration with the aid of molecular modeling.
Journal of Medicinal Chemistry
59
(6)
, pp. 2688-2703.
10.1021/acs.jmedchem.5b01935
|
|
|
Nannetti, Giulio ORCID: https://orcid.org/0000-0003-3227-1537, Pagni, Silvana, Parisi, Saverio G., Alberti, Alfredo, Loregian, Arianna and Palù, Giorgio
2016.
Development of a simple HPLC-UV method for the determination of the hepatitis C virus inhibitor simeprevir in human plasma.
Journal of Pharmaceutical and Biomedical Analysis
121
, pp. 197-203.
10.1016/j.jpba.2016.01.019
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Mercorelli, Beatrice, Luganini, Anna, Nannetti, Giulio ORCID: https://orcid.org/0000-0003-3227-1537, Tabarrini, Oriana, Palù, Giorgio, Gribaudo, Giorgio and Loregian, Arianna
2016.
Drug repurposing approach identifies inhibitors of the prototypic viral transcription Factor IE2 that block human cytomegalovirus replication.
Cell Chemical Biology
23
(3)
, pp. 340-351.
10.1016/j.chembiol.2015.12.012
|
|
|
Massari, Serena, Nannetti, Giulio ORCID: https://orcid.org/0000-0003-3227-1537, Desantis, Jenny, Muratore, Giulia, Sabatini, Stefano, Manfroni, Giuseppe, Mercorelli, Beatrice, Cecchetti, Violetta, Palù, Giorgio, Cruciani, Gabriele, Loregian, Arianna, Goracci, Laura and Tabarrini, Oriana
2015.
A broad anti-influenza hybrid small molecule that potently disrupts the interaction of polymerase acidic protein-basic protein 1 (PA-PB1) subunits.
Journal of Medicinal Chemistry
58
(9)
, pp. 3830-3842.
10.1021/acs.jmedchem.5b00012
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|
|
Loregian, Arianna, Mercorelli, Beatrice, Nannetti, Giulio ORCID: https://orcid.org/0000-0003-3227-1537, Compagnin, Chiara and Palù, Giorgio
2014.
Antiviral strategies against influenza virus: towards new therapeutic approaches.
Cellular and Molecular Life Sciences
71
(19)
, pp. 3659-3683.
10.1007/s00018-014-1615-2
|
|
|
Lepri, Susan, Nannetti, Giulio ORCID: https://orcid.org/0000-0003-3227-1537, Muratore, Giulia, Cruciani, Gabriele, Ruzziconi, Renzo, Mercorelli, Beatrice, Palù, Giorgio, Loregian, Arianna and Goracci, Laura
2014.
Optimization of small-molecule inhibitors of influenza virus polymerase: From thiophene-3-carboxamide to polyamido scaffolds.
Journal of Medicinal Chemistry
57
(10)
, pp. 4337-4350.
10.1021/jm500300r
|
|
|
Massari, Serena, Nannetti, Giulio ORCID: https://orcid.org/0000-0003-3227-1537, Goracci, Laura, Sancineto, Luca, Muratore, Giulia, Sabatini, Stefano, Manfroni, Giuseppe, Mercorelli, Beatrice, Cecchetti, Violetta, Facchini, Marzia, Palù, Giorgio, Cruciani, Gabriele, Loregian, Arianna and Tabarrini, Oriana
2013.
Structural investigation of Cycloheptathiophene-3-carboxamide derivatives targeting influenza virus polymerase assembly.
Journal of Medicinal Chemistry
56
(24)
, pp. 10118-10131.
10.1021/jm401560v
|
|
|
Saladini, Francesco, Foley, Brian T., Rosi, Andrea, Vicenti, Ilaria, Nannetti, Giulio ORCID: https://orcid.org/0000-0003-3227-1537, Meini, Genny, Razzolini, Francesca and Zazzi, Maurizio
2012.
Near full-length sequence analysis of HIV Type 1 BF recombinants from Italy.
AIDS Research and Human Retroviruses
28
(3)
, p. 299.
10.1089/aid.2011.0002
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