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Number of items: 114.

A

Abdurazova, P.A., Nazarbek, U.B., Bolysbek, A.A., Sarypbekova, N.K., Kenzhibayeva, G.S., Kambarova, G.A., Sataev, M.S., Koshkarbaeva, Sh.T., Tleuova, A.B., Perni, Stefano and Prokopovich, Polina

2017. Preparation of photochemical coatings of metal films (copper, silver and gold) on dielectric surfaces and studying their antimicrobial properties. Colloids and Surfaces A: Physicochemical and Engineering Aspects 532 , pp. 63-69. 10.1016/j.colsurfa.2017.06.070

Ahmad, Nisar, Subhan, Fazal, Islam, Nazar Ur, Shahid, Muhammed, Rahman, Faiz Ur and Sewell, Robert D. E. 2017. Gabapentin and its salicylaldehyde derivative alleviate allodynia and hypoalgesia in a cisplatin-induced neuropathic pain model. European Journal of Pharmacology 814 , pp. 302-312. 10.1016/j.ejphar.2017.08.040

Akbar, s, Subhan, F, Karim, N, Aman, U, Ullah, S, Shahid, M, Ahmad, N, Fawad, K and Sewell, Robert 2017. Characterization of 6-methoxyflavanone as a novel anxiolytic agent: A behavioral and pharmacokinetic approach. European Journal of Pharmacology 801 , pp. 19-27. 10.1016/j.ejphar.2017.02.047

Al Thaher, Yazan, Perni, Stefano and Prokopovich, Polina

2017. Nano-carrier based drug delivery systems for sustained antimicrobial agent release from orthopaedic cementous material. Advances in Colloid and Interface Science 249 , pp. 234-247. 10.1016/j.cis.2017.04.017

Alam, Javaid, Subhan, Fazal, Ullah, Ihsan, Shahid, Muhammad, Ali, Gowhar and Sewell, Robert David Edmund 2017. Synthetic and natural antioxidants attenuate cisplatin-induced vomiting. BMC Pharmacology and Toxicology 18 (4) 10.1186/s40360-016-0110-9

AlAmri, Mubarak A., Kadri, Hachemi, Dhiani, Binar Asrining, Mahmood, Shumail, Elzwawi, Abdulrahman and Mehellou, Youcef

2017. WNK-signaling inhibitors as potential new antihypertensive drugs. Chemmedchem 10.1002/cmdc.201700425

Alamri, Mubarak A., Kadri, Hachemi, Alderwick, Luke J., Simpkins, Nigel S. and Mehellou, Youcef

2017. Rafoxanide and Closantel inhibit SPAK and OSR1 kinases by binding to a highly conserved allosteric site on their C-terminal domains. ChemMedChem 12 (9) , pp. 639-645. 10.1002/cmdc.201700077

Aldrovandi, MacEler, Hinz, Christine, Lauder, Sarah N, Podmore, Helen, Hornshaw, Martin, Slatter, David A, Tyrrell, Victoria J, Clark, Stephen R, Marnett, Lawrence J., Collins, Peter W

, Murphy, Robert C and O'Donnell, Valerie B

2017. DioxolaneA3-phosphatidylethanolamines are generated by human platelets and stimulate neutrophil integrin expression. Redox Biology 11 , pp. 663-672. 10.1016/j.redox.2017.01.001

Ali, Faraz Mahmood, Kay, Richard, Finlay, Andrew Yule

, Piguet, Vincent, Kupfer, Joerg, Dalgard, Florence and Salek, M. Sam 2017. Mapping of the DLQI scores to EQ-5D utility values using ordinal logistic regression. Quality of Life Research 26 , pp. 3025-3034. 10.1007/s11136-017-1607-4

Alsaqati, Mouhamed, Thomas, Rhian S. and Kidd, Emma

2017. Proteins involved in endocytosis are upregulated by ageing in the normal human brain: implications for the development of Alzheimer's disease. Journals of Gerontology, Series A 73 (3) , pp. 289-298. 10.1093/gerona/glx135

Ayaz, Muhammad, Subhan, Fazal, Sadiq, Abdul, Ullah, Farhat, Ahmed, Jawad and Sewell, Robert David Edmund 2017. Cellular efflux transporters and the potential role of natural products in combating efflux mediated drug resistance. Frontiers in Bioscience 22 (4) , pp. 732-756. 10.2741/4513

B

Bassetto, Marcella

, Ferla, Salvatore

, Giancotti, Gilda, Pertusati, Fabrizio

, Westwell, Andrew D.

, Brancale, Andrea

and McGuigan, Christopher 2017. Rational design and synthesis of novel phenylsulfonyl-benzamides as anti-prostate cancer agents. MedChemComm 8 (7) , pp. 1414-1420. 10.1039/C7MD00164A

Bassetto, Marcella

, Leyssen, Pieter, Neyts, Johan, Yerukhimovich, Mark M., Frick, David N. and Brancale, Andrea

2017. Shape-based virtual screening, synthesis and evaluation of novel pyrrolone derivatives as antiviral agents against HCV. Bioorganic & Medicinal Chemistry Letters 27 (4) , pp. 936-940. 10.1016/j.bmcl.2016.12.087

Bassetto, Marcella

, Leyssen, Pieter, Neyts, Johan, Yerukhimovich, Mark M., Frick, David N., Courtney-Smith, Matthew and Brancale, Andrea

2017. In silico identification, design and synthesis of novel piperazine-based antiviral agents targeting the hepatitis C virus helicase. European Journal of Medicinal Chemistry 125 , pp. 1115-1131. 10.1016/j.ejmech.2016.10.043

Baxani Kamal, Divesh 2017. Hydrogel encapsulated droplet interface bilayer networks as a chassis for artificial cells and a platform for membrane studies. PhD Thesis, Cardiff University.

Item availability restricted.

Baxani Kamal, Divesh, Morgan, A. J., Li, J.

, Barrow, D. A.

and Castell, Oliver

2017. The microfluidic manufacture of encapsulated droplet interface bilayers using a hybrid 3D-printed coaxial device. Presented at: 20th International Conference on Miniaturized Systems for Chemistry and Life Sciences (MicroTAS 2016), Dublin, Ireland, 9-13 October 2016. Proceedings of the 20th International Conference on Miniaturized Systems for Chemistry and Life Sciences (MicroTAS 2016). Red Hook, New York: Curran Associates, Inc.,

Brancale, Andrea

, Shailubhai, Kunwar, Ferla, Salvatore

, Ricci, Antonio, Bassetto, Marcella

and Jacob, Gary S. 2017. Therapeutically targeting guanylate cyclase-C: computational modeling of plecanatide, a uroguanylin analog. Pharmacology Research & Perspectives 5 (2) , e00295. 10.1002/prp2.295

Brazzale, C., Mastrotto, F., Moody, P., Watson, P. D.

, Balasso, A., Malfanti, A., Mantovani, G., Caliceti, P., Alexander, C., Jones, A. T.

and Salmaso, S. 2017. Control of targeting ligand display by pH-responsive polymers on gold nanoparticles mediates selective entry into cancer cells. Nanoscale 9 (31) , pp. 11137-11147. 10.1039/C7NR02595E

Breger, Ludivine S., Kienle, Korbinian, Smith, Gaynor A.

, Dunnett, Stephen B.

and Lane, Emma L.

2017. Influence of chronic L-DOPA treatment on immune response following allogeneic and xenogeneic graft in a rat model of Parkinson's disease. Brain, Behavior, and Immunity 61 , pp. 155-164. 10.1016/j.bbi.2016.11.014

C

Campbell, Anthony 2017. Fundamentals of Intracellular Calcium. Wiley-Blackwell.

Cavaliere, Alessandra, Probst, Katrin, Westwell, Andrew

and Slusarczyk, Magdalena

2017. Fluorinated nucleosides as an important class of anticancer and antiviral agents. Future Medicinal Chemistry 9 (15)

Chen, Hung-Chang, Joalland, Noémie, Bridgeman, John S, Alchami, Fouad S, Jarry, Ulrich, Khan, Mohd Wajid A, Piggott, Luke, Shanneik, Yasmin, Li, Jianqiang, Herold, Marco J, Herrmann, Thomas, Price, David A.

, Gallimore, Awen M.

, Clarkson, Richard W.

, Scotet, Emmanuel, Moser, Bernhard

and Eberl, Matthias

2017. Synergistic targeting of breast cancer stem-like cells by human γδ T cells and CD8+ T cells. Immunology and Cell Biology 95 (7) , pp. 620-629. 10.1038/icb.2017.21

Cima, Cecilia 2017. Computer-aided design and synthesis of novel anti-DENV nucleoside analogues. PhD Thesis, Cardiff University.

Item availability restricted.

Courtenay, Molly

, Khanfer, Riyad, Harries-Huntly, Gail, Deslandes, Rhian

, Gillespie, David, Hodson, Karen

, Morris, Gary, Pritchard, Anthony and Williams, Elizabeth 2017. Overview of the uptake and implementation of non-medical prescribing in Wales: a national survey. BMJ Open 7 (9) , e015313. 10.1136/bmjopen-2016-015313

Courtenay, Molly

, Rowbotham, Samantha, Lim, Rosemary, Deslandes, Rhian

, Hodson, Karen

, MacClure, Katie, Peters, Sarah and Stewart, Derek 2017. Antibiotics for acute respiratory tract infections: a mixed-methods study of patient experiences of non-medical prescriber management. BMJ Open 7 (3) , e013515. 10.1136/bmjopen-2016-013515

D

Derudas, Marco, Vanpouille, Christophe, Carta, Davide, Zicari, Sonia, Andrei, Graciela, Snoeck, Robert, Brancale, Andrea

, Margolis, Leonid, Balzarini, Jan and McGuigan, Christopher

2017. Virtual screening of acyclovir derivatives as potential antiviral agents: design, synthesis, and biological evaluation of new acyclic nucleoside protides. Journal of Medicinal Chemistry 60 (18) , pp. 7876-7896. 10.1021/acs.jmedchem.7b01009

Desantis, Jenny, Nannetti, Giulio

, Massari, Serena, Barreca, Maria Letizia, Manfroni, Giuseppe, Cecchetti, Violetta, Palù, Giorgio, Goracci, Laura, Loregian, Arianna and Tabarrini, Oriana 2017. Exploring the cycloheptathiophene-3-carboxamide scaffold to disrupt the interactions of the influenza polymerase subunits and obtain potent anti-influenza activity. European Journal of Medicinal Chemistry 138 , pp. 128-139. 10.1016/j.ejmech.2017.06.015

Dul, M.

, Stefanidou, M.., Porta, P., Serve, J., O'Mahony, C., Malissen, B., Henri, S., Levin, Y., Kochba, E., Wong, F.S.

, Dayan, C.

, Coulman, S.A.

and Birchall, J.C.

2017. Hydrodynamic gene delivery in human skin using a hollow microneedle device. Journal of Controlled Release 265 , pp. 120-131. 10.1016/j.jconrel.2017.02.028

E

Ehrhardt, Carsten, Bäckman, Per, Couet, William, Edwards, Chris, Forbes, Ben, Fridén, Markus, Gumbleton, Mark

, Hosoya, Ken-Ichi, Kato, Yukio, Nakanishi, Takeo, Takano, Mikihisa, Terasaki, Tetsuya and Yumoto, Ryoko 2017. Current progress toward a better understanding of drug disposition within the lungs: summary proceedings of the first workshop on drug transporters in the lungs. Journal of Pharmaceutical Sciences 106 (9) , pp. 2234-2244. 10.1016/j.xphs.2017.04.011

Elabi, Osama 2017. The effect of L-dopa and neuroprotective agents on cell replacement therapy for Parkinson’s disease. PhD Thesis, Cardiff University.

Item availability restricted.

Elbaramawi, Samar S., Ibrahim, Samy M., Lashine, El-Sayed M., El-Sadek, Mohamed E., Mantzourani, Efi

and Simons, Claire

2017. Exploring the binding sites of Staphylococcus aureus phenylalanine tRNA synthetase: A homology model approach. Journal of Molecular Graphics and Modelling 73 , pp. 36-47. 10.1016/j.jmgm.2017.02.002

Elsadig, Hwaida, Weiss, Marjorie

, Scott, Jenny and Laaksonen, Raisa 2017. Exploring the challenges for clinical pharmacists in Sudan. International Journal of Clinical Pharmacy 39 (5) , pp. 1047-1054. 10.1007/s11096-017-0521-8

F

Famiglini, Valeria, La Regina, Giuseppe, Coluccia, Antonio, Masci, Domiziana, Brancale, Andrea

, Badia, Roger, Riveira Muñoz, Eva, Este, Jose A., Crespan, Emmanuele, Brambilla, Alessandro, Maga, Giovanni, Catalano, Myriam, Limatola, Cristina, Formica, Francesca Romana Romana, Cirilli, Roberto, Novellino, Ettore and Silvestri, Romano 2017. Chiral indolylarylsulfone non-nucleoside reverse transcriptase inhibitors as new potent and broad spectrum anti-HIV-1 agents. Journal of Medicinal Chemistry 60 (15) , pp. 6528-6547. 10.1021/acs.jmedchem.6b01906

G

Gao, Yongsheng, Newland, Ben

, Zhou, Dezhong, Matyjaszewski, Krzysztof and Wang, Wenxin 2017. Controlled polymerization of multivinyl monomers: Formation of cyclized/knotted single-chain polymer architectures. Angewandte Chemie International Edition 56 (2) , pp. 450-460. 10.1002/anie.201608786

NuCana Biomed Ltd 2017. Adenosine derivatives for use in the treatment of cancer. WO2017207989A1. [Patent].

Grisley, Lauren, Manning, Abigail, Lee, Harry, McRae, David, Williams, Emma and Mantzourani, Efthymia

2017. Evaluation of the Cwm Taf University Health Board Domiciliary Medicines Use Review (Dom-MUR) Service. Global Journal of Pharmacy & Pharmaceutical Sciences 1 (4) , .555567.

Gruden, M. A, Davydova, T. V, Fomina, V. G, Vetrile, L. A, Morozova-Roche, L. A and Sewell, Robert 2017. Antibodies to glutamate reversed the amnesic effects of proinflammatory S100A9 protein fibrils in aged C57Bl/6 mice. Bulletin of Experimental Biology and Medicine 162 (4) , pp. 430-432. 10.1007/s10517-017-3632-2

Guelfi, Gabriella, Stefanetti, Valentina, Zampini, Danilo, Oommen, Oommen P.

, Breccia, Gabriele, Dall'Aglio, Cecilia, Arcelli, Rolando, Cochetti, Giovanni, Boni, Andrea and Mearini, Ettore 2017. Gold nanoparticles approach to detect chondroitin sulphate and hyaluronic acid urothelial coating. Scientific Reports 7 (1) , 10355. 10.1038/s41598-017-09872-0

H

Hamdy, Rania, Ziedan, Noha, Ali, Samina, Bordoni, Cinzia, El-Sadek, Mohamed, Lashin, Elsaid, Brancale, Andrea

, Jones, Arwyn Tomos

and Westwell, Andrew D

2017. Synthesis and evaluation of 5-(1H-indol-3-yl)-N-aryl-1,3,4-oxadiazol-2-amines as Bcl-2 inhibitory anticancer agents. Bioorganic & Medicinal Chemistry Letters 27 (4) , pp. 1037-1040. 10.1016/j.bmcl.2016.12.061

Hendriks, Hans R, Govaerts, Anne-Sophie, Fichtner, Iduna, Burtles, Sally, Westwell, Andrew

and Peters, Godefridus J 2017. Pharmacologically directed strategies in academic anticancer drug discovery based on the European NCI compounds initiative. British Journal of Cancer 117 , pp. 195-202. 10.1038/bjc.2017.167

Houston, David M. J., Bugert, Joachim J.

, Denyer, Stephen P. and Heard, Charles M.

2017. Potentiated virucidal activity of pomegranate rind extract (PRE) and punicalagin against Herpes simplex virus (HSV) when co-administered with zinc (II) ions, and antiviral activity of PRE against HSV and aciclovir-resistant HSV. PLoS ONE 12 (6) , e0179291. 10.1371/journal.pone.0179291

Houston, David M. J., Robins, Bethan, Bugert, Joachim J., Denyer, Stephen P. and Heard, Charles M.

2017. In vitro permeation and biological activity of punicalagin and zinc (II) across skin and mucous membranes prone to Herpes simplex virus infection. European Journal of Pharmaceutical Sciences 96 , pp. 99-106. 10.1016/j.ejps.2016.08.013

Houston, David, Bugert, Joachim

, Denyer, Stephen P. and Heard, Charles M.

2017. Anti-inflammatory activity of Punica granatum L. (Pomegranate) rind extracts applied topically to ex vivo skin. European Journal of Pharmaceutics and Biopharmaceutics 112 , pp. 30-37. 10.1016/j.ejpb.2016.11.014

J

James, Edward, Pertusati, Fabrizio

, Brancale, Andrea

and McGuigan, Christopher

2017. Kinase-independent phosphoramidate S1P1 receptor agonist benzyl ether derivatives. Biorganic and Medicinal Chemistry Letters 27 (6) , pp. 1371-1378. 10.1016/j.bmcl.2017.02.011

James, Edward 2017. Phosphorus prodrugs of S1P receptor modulators as a novel therapeutic opportunity. PhD Thesis, Cardiff University.

Item availability restricted.

Jimenez Antunez, Carmen

2017. Design, synthesis and biological evaluation of nucleoside phosphoramidates with potential anticancer activity. PhD Thesis, Cardiff University.

Item availability restricted.

Jonas, Kim C., Melrose, Timothy, Thompson, Iain R., Baxter, Gary Francis

, Lipscomb, Victoria J., Niessen, Stijn J., Lawson, Charlotte, McArdle, Craig A., Roberson, Mark S., McGonnell, Imelda M., Wheeler-Jones, Caroline P. and Fowkes, Robert C. 2017. Natriuretic peptide activation of extracellular regulated kinase 1/2 (ERK1/2) pathway by particulate guanylyl cyclases in GH3 somatolactotropes. Cell and Tissue Research 369 (3) , pp. 567-578. 10.1007/s00441-017-2624-x

Jones, Samuel Rhys 2017. Exploring Focal Adhesion Kinase (FAK) as a therapeutic target in triple negative breast cancer. PhD Thesis, Cardiff University.

Item availability restricted.

Jones, Brian, Ecenarro, Susana, Whiteside, Ben, Birchall, James

and Coulman, Sion

2017. Imaging techniques for dry powder inhaler capsules. Inhalation

Joshi, Lovleen Tina, Welsch, Angelina, Hawkins, Jennifer and Baillie, Les

2017. The effect of hospital biocide sodium dichloroisocyanurate on the viability and properties of Clostridium difficile spores. Letters in Applied Microbiology 65 (3) , pp. 199-205. 10.1111/lam.12768

K

Kadri, Hachemi, Alamri, Mubarak A., Navratilova, Iva H., Alderwick, Luke J., Simpkins, Nigel S. and Mehellou, Youcef

2017. Towards the development of small molecule MO25-binders as potential indirect SPAK/OSR1 kinase inhibitors. ChemBioChem 18 (5) , pp. 460-465. 10.1002/cbic.201600620

Karwi, Qutuba G., Bornbaum, Julia, Boengler, Kerstin, Torregrossa, Roberta, Whiteman, Matthew, Wood, Mark E., Schulz, Rainer and Baxter, Gary F.

2017. Ap39, a mitochondria-targeting hydrogen sulfide (H2 s) donor, protects against myocardial reperfusion injury independently of salvage kinase signalling. British Journal of Pharmacology 174 (4) , pp. 287-301. 10.1111/bph.13688

Kedge, Jonathan L., Nguyen, Huy V., Khan, Zahra, Male, Louise, Hodges, Media K. Ismail Holly V. Roberts Ni, Horswell, Sarah L., Mehellou, Youcef

and Tucker, James H. R. 2017. Organometallic nucleoside analogues: effect of hydroxyalkyl linker length on cancer cell line toxicity. European Journal of Inorganic Chemistry 2017 (2) , pp. 466-476. 10.1002/ejic.201600853

Khmaladze, E, Su, W, Zghenti, E, Buyuk, F, Sahin, M, Nicolich,MP, MP, Baillie, Les

, Obiso, R and Kotorashvili, A 2017. Molecular genotyping of bacillus anthracis strains from Georgia and northeastern part of Turkey. Journal of Bacteriology and Mycology 4 (3)

Kjos, Ingrid, Borg Distefano, Marita, Sætre, Frank, Repnik, Urska, Holland, Petter, Jones, Arwyn T.

, Engedal, Nikolai, Simonsen, Anne, Bakke, Oddmund and Progida, Cinzia 2017. Rab7b modulates autophagic flux by interacting with Atg4B. EMBO reports 18 (10) , pp. 1727-1739. 10.15252/embr.201744069

L

La Regina, Giuseppe, Bai, Ruoli, Coluccia, Antonio, Famiglini, Valeria, Passacantilli, Sara, Naccarato, Valentina, Ortar, Giorgio, Mazzoccoli, Carmela, Ruggieri, Vitalba, Agriesti, Francesca, Piccoli, Claudia, Tataranni, Tiziana, Nalli, Marianna, Brancale, Andrea

, Vultaggio, Stefania, Mercurio, Ciro, Varasi, Mario, Saponaro, Concetta, Sergio, Sara, Maffia, Michele, Coluccia, Addolorata Maria Luce, Hamel, Ernest and Silvestri, Romano 2017. 3-Aroyl-1,4-diarylpyrroles inhibit chronic myeloid leukemia cell growth through an interaction with tubulin. ACS Medicinal Chemistry Letters 8 (5) , pp. 521-526. 10.1021/acsmedchemlett.7b00022

Lauder, Sarah N., Allen-Redpath, Keith, Slatter, David A., Aldrovandi, Maceler, O'Connor, Anne, Farewell, Daniel

, Percy, Charles L., Molhoek, Jessica E., Rannikko, Sirpa, Tyrrell, Victoria J., Ferla, Salvatore

, Milne, Ginger L., Poole, Alastair W., Thomas, Christopher P.

, Obaji, Samya, Taylor, Philip R., Jones, Simon A.

, deGroot, Philip G., Urbanus, Rolf T., Horkko, Sohvi, Uderhardt, Stefan, Ackermann, Jochen, Jenkins, P. Vince, Brancale, Andrea

, Kronke, Gerhard, Collins, Peter W.

and O'Donnell, Valerie B.

2017. Networks of enzymatically oxidized membrane lipids support calcium-dependent coagulation factor binding to maintain hemostasis. Science Signaling 10 (507) , eaan2787. 10.1126/scisignal.aan2787

Li, J.

, Baxani Kamal, Divesh, Castell, Oliver

and Barrow, David

2017. Formation of chemically responsive multisomes using droplet microfluidics. Presented at: 20th International Conference on Miniaturized Systems for Chemistry and Life Sciences (MicroTAS 2016), Dublin, Ireland, 9-13 October 2016. Proceedings of the 20th International Conference on Miniaturized Systems for Chemistry and Life Sciences (MicroTAS 2016). Red Hook, NY: Curran Associates, Inc.,

Lowe, Alexander P. P., Thomas, Rhian S., Nials, Anthony T., Kidd, Emma J.

, Broadley, Kenneth J.

and Ford, William R.

2017. Route of administration affects corticosteroid sensitivity of a combined ovalbumin and lipopolysaccharide model of asthma exacerbation in guinea-pigs. Journal of Pharmacology and Experimental Therapeutics 362 (2) , pp. 327-337. 10.1124/jpet.117.241927

Lymperatou, Dionysia

2017. Exploring the impact of anti-oestrogen resistance on the capacity of breast cancer cells to modulate bone cell function and their sensitivity to bisphosphonates. PhD Thesis, Cardiff University.

Item availability restricted.

M

Mantzourani, Efthymia

, Potter Floyd, Georgia and James, Delyth 2017. Pharmacy students' reflections on a 'mock medicines' activity: Exploring intentional and unintentional nonadherence. Pharmacy Education 17 (1) , pp. 1-7.

Mantzourani, Efthymia

, Way, Cheryl and Hodson, Karen

2017. Does an integrated information technology system provide support for community pharmacists undertaking discharge medicines reviews? An exploratory study. Integrated Pharmacy Research and Practice 6 , pp. 145-156.

Martin, Christopher, Alcock, Natalie, Hiom, Sarah and Birchall, James C.

2017. Development and evaluation of topical gabapentin formulations. Pharmaceutics 9 (3) , p. 31. 10.3390/pharmaceutics9030031

Mashaki, Emel 2017. Evaluation of the regulatory review system in Turkey and the development of a new model for improving the approval process. PhD Thesis, Cardiff University.

Item availability restricted.

Massari, Serena, Desantis, Jenny, Nannetti, Giulio

, Sabatini, Stefano, Tortorella, Sara, Goracci, Laura, Cecchetti, Violetta, Loregian, Arianna and Tabarrini, Oriana 2017. Efficient and regioselective one-step synthesis of 7-aryl-5-methyl- and 5-aryl-7-methyl-2-amino-[1,2,4]triazolo[1,5-a]pyrimidine derivatives. Organic and Biomolecular Chemistry 15 (37) , pp. 7944-7955. 10.1039/C7OB02085F

McGrath, Marie, Coulman, Sion

, Birchall, James C.

and Prausnitz, Mark 2017. Editorial. Journal of Controlled Release 265 , p. 1. 10.1016/j.jconrel.2017.10.030

Mikhail, Ashraf, Brown, Christopher, Williams, Jennifer Ann, Mathrani, Vinod, Shrivastava, Rajesh, Evans, Jonathan, Isaac, Hayleigh and Bhandari, Sunil 2017. Renal association clinical practice guideline on anaemia of chronic kidney disease. BMC Nephrology 18 (1) , 345. 10.1186/s12882-017-0688-1

Moreno, Esther, Schwartz, Juana, Calvo, Alba, Blanco, Laura, Larrea, Esther, Irache, Juan M, Sanmartín, Carmen, Coulman, Sion A

, Soto, Manuel, Birchall, James C

and Espuelas, Socorro 2017. Skin vaccination using microneedles coated with a plasmid DNA cocktail encoding nucleosomal histones of Leishmania spp. International Journal of Pharmaceutics 533 (1) , pp. 236-244. 10.1016/j.ijpharm.2017.09.055

Moriconi, Chiara

, Palmieri, Valentina, di Santo, Riccardo, Tornillo, Giusy, Papi, Massimiliano, Pilkington, Geoff, De Spirito, Marco and Gumbleton, Mark

2017. INSIDIA: a FIJI macro delivering high-throughput and high-content spheroid invasion analysis. Biotechnology Journal 12 (10) , 1700140. 10.1002/biot.201700140

Moriconi, Chiara

, Palmieri, Valentina, Tornillo, Giusy, Fillmore, Helen, Pilkington, Geoff and Gumbleton, Mark

2017. Caveolin-1 implicated as a pro-invasive gene in high-grade glioma cell models: implementation of a 3d spheroid matrix invasion assay. Neuro-Oncology 19 (S1) , i21-i22. 10.1093/neuonc/now293.080

Morris, Christopher J., Aljayyoussi, Ghaith, Mansour, Omar, Griffiths, Peter and Gumbleton, Mark

2017. Endocytic uptake, transport and macromolecular interactions of anionic PAMAM dendrimers within lung tissue. Pharmaceutical Research 34 (12) , pp. 2517-2531. 10.1007/s11095-017-2190-7

Morrison, Peter

, Porfiryeva, Natalia N, Chahal, Sukhmanpreet, Salakhov, Ilgiz A., Lacourt, Charlene, Semina, Irina I, Moustafine, Rouslan I. and Khutoryanskiy, Vitaliy V. 2017. Crown Ethers: novel permeability enhancers for ocular drug delivery? Molecular Pharmaceutics 14 (10) , pp. 3528-3538. 10.1021/acs.molpharmaceut.7b00556

N

Nannetti, Giulio

, Messa, Lorenzo, Celegato, Marta, Pagni, Silvana, Basso, Monica, Parisi, Saverio G., Palù, Giorgio and Loregian, Arianna 2017. Development and validation of a simple and robust HPLC method with UV detection for quantification of the hepatitis C virus inhibitor daclatasvir in human plasma. Journal of Pharmaceutical and Biomedical Analysis 134 , pp. 275-281. 10.1016/j.jpba.2016.11.032

Netzler, Natalie E., Enosi Tuipulotu, Daniel, Eltahla, Auda A., Lun, Jennifer H., Ferla, Salvatore

, Brancale, Andrea

, Urakova, Nadya, Frese, Michael, Strive, Tanja, Mackenzie, Jason M. and White, Peter A. 2017. Broad-spectrum non-nucleoside inhibitors for caliciviruses. Antiviral Research 146 , pp. 65-75. 10.1016/j.antiviral.2017.07.014

Neusser, G., Eppler, S., Bowen, J.

, Allender, C. J., Walther, P., Mizaikoff, B. and Kranz, C. 2017. FIB and MIP: understanding nanoscale porosity in molecularly imprinted polymers via 3D FIB/SEM tomography. Nanoscale 9 (38) , pp. 14327-14334. 10.1039/C7NR05725C

Newland, Benjamin

, Baeger, Marcel, Eigel, Dimitri, Newland, Heike and Werner, Carsten 2017. Oxygen-producing gellan gum hydrogels for dual delivery of either oxygen or peroxide with doxorubicin. ACS Biomaterials Science & Engineering 3 (5) , pp. 787-792. 10.1021/acsbiomaterials.7b00078

Nimmanon, T., Ziliotto, S., Morris, S., Flanagan, L. and Taylor, K. M.

2017. Phosphorylation of zinc channel ZIP7 drives MAPK, PI3K and mTOR growth and proliferation signalling. Metallomics 9 (5) , pp. 471-481. 10.1039/C6MT00286B

O

Osgerby, Laura, Lai, Yu-Chiang, Thornton, Peter J., Amalfitano, Joseph, Le Duff, Cécile S., Jabeen, Iqra, Kadri, Hachemi, Miccoli, Ageo, Tucker, James H. R., Muqit, Miratul M. K. and Mehellou, Youcef

2017. Kinetin riboside and its ProTides activate the Parkinson's Disease associated PTEN-Induced Putative Kinase 1 (PINK1) independent of mitochondrial depolarization. Journal of Medicinal Chemistry 60 (8) , pp. 3518-3524. 10.1021/acs.jmedchem.6b01897

P

Parmeggiani, F

and Huang, P 2017. Designing repeat proteins. Current Opinion in Structural Biology 45 (8) , pp. 116-123. 10.1016/j.sbi.2017.02.001

Paul, Graham R. 2017. Defining dosimetry and implications for aerosol presentation for non-clinical development of respiratory drugs. PhD Thesis, Cardiff University.

Item availability restricted.

Paul, Graham, Gumbleton, Mark

and Somers, Graham I 2017. Effect of conditioning on rat lung function measurements and implications for exposure and dose estimation of inhaled drugs. Inhalation

Perni, Stefano and Prokopovich, Polina

2017. Poly-beta-amino-esters nano-vehicles based drug delivery system for cartilage. Nanomedicine: Nanotechnology, Biology and Medicine 13 (2) , pp. 539-548. 10.1016/j.nano.2016.10.001

Pertusati, Fabrizio

, Nutz, Eva, Kariuki, Benson

and Coogan, Michael P. 2017. Synthesis and substrate-controlled reactions of 2,2′-unsaturated biquinazolinones. Tetrahedron 73 (1) , pp. 55-63. 10.1016/j.tet.2016.11.060

Pertusati, Fabrizio

, Serafini, Sara, Albadry, Najmiyah, Snoeck, Robert and Andrei, Graciela 2017. Phosphonoamidate prodrugs of C5-substituted pyrimidine acyclic nucleosides for antiviral therapy. Antiviral Research 143 , pp. 262-268. 10.1016/j.antiviral.2017.04.013

Preedy, Emily Callard, Perni, Stefano and Prokopovich, Polina

2017. Cobalt and titanium nanoparticles influence on mesenchymal stem cell elasticity and turgidity. Colloids and Surfaces B: Biointerfaces 157 , pp. 146-156. 10.1016/j.colsurfb.2017.05.019

Price, Daniel F., Luscombe, Chris N., Eddershaw, Peter J., Edwards, Chris D. and Gumbleton, Mark

2017. The differential absorption of a series of P-glycoprotein substrates in isolated perfused lungs from Mdr1a/1b genetic knockout mice can be attributed to distinct physico-chemical properties: an insight into predicting transporter-mediated, pulmonary specific disposition. Pharmaceutical Research 34 (12) , pp. 2498-2516. 10.1007/s11095-017-2220-5

R

Roberts-Dalton, H. D.

, Cocks, A., Falcon-Perez, J. M., Sayers, E. J.

, Webber, J. P.

, Watson, P.

, Clayton, A.

and Jones, A. T.

2017. Fluorescence labelling of extracellular vesicles using a novel thiol-based strategy for quantitative analysis of cellular delivery and intracellular traffic. Nanoscale 9 (36) , pp. 13693-13706. 10.1039/C7NR04128D

Roberts-Dalton, Hope

2017. Defining endocytic pathways to characterise the cellular uptake of extracellular vesicles. PhD Thesis, Cardiff University.

Item availability restricted.

Romagnoli, Romeo, Baraldi, Pier Giovanni, Prencipe, Filippo, Oliva, Paola, Baraldi, Stefania, Salvador, Maria Kimatrai, Lopez-Cara, Luisa Carlota, Brancale, Andrea

, Ferla, Salvatore

, Hamel, Ernest, Ronca, Roberto, Bortolozzi, Roberta, Mariotto, Elena, Porcù, Elena, Basso, Giuseppe and Viola, Giampietro 2017. Synthesis and Biological Evaluation of 2-Methyl-4,5-Disubstituted Oxazoles as a Novel Class of Highly Potent Antitubulin Agents. Scientific Reports 7 , 46356. 10.1038/srep46356

Roshanbinfar, Kaveh, Hilborn, Jöns, Varghese, Oommen P. and Oommen, Oommen P.

2017. Injectable and thermoresponsive pericardial matrix derived conductive scaffold for cardiac tissue engineering. RSC Adv. 7 , pp. 31980-31988. 10.1039/C7RA03780E

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Salim, Mahboob, Knowles, Timothy J., Baker, Alfie T., Davey, Martin S., Jeeves, Mark, Sridhar, Pooja, Wilkie, John, Willcox, Carrie R., Kadri, Hachemi, Taher, Taher E, Vantourout, Pierre, Hayday, Adrian, Mehellou, Youcef

, Mohammed, Fiyaz and Willcox, Benjamin E. 2017. BTN3A1 discriminates γδ T cell phosphoantigens from non-antigenic small molecules via a conformational sensor in its B30.2 domain. ACS Chemical Biology 12 (10) , pp. 2631-2643. 10.1021/acschembio.7b00694

Sataev, M. S., Abdurasova, P. A., Koshkarbaeva, Sh. T., Bolisbek, A. A., Saripbekova, N. K., Kambarova, G. A., Koblanova, O. N., Perni, S. and Prokopovich, Polina

2017. A low-temperature gold coating of the dielectric surfaces employing phosphine gas as a reducing agent. Colloids and Surfaces A: Physicochemical and Engineering Aspects 521 , pp. 86-91. 10.1016/j.colsurfa.2016.11.029

Scott, Hannah

2017. Extracellular microRNAs as messengers in the central and peripheral nervous system. Neuronal Signaling 1 (4) , NS20170112. 10.1042/NS20170112

Serpi, Michaela

, De Biasi, Roberto, Pertusati, Fabrizio

, Slusarczyk, Magdalena

and McGuigan, Christopher 2017. Synthetic approaches for the preparation of phosphoramidate prodrugs of 2’-deoxypseudoisocytidine. ChemistryOpen 6 (3) , pp. 424-436. 10.1002/open.201700019

Shahid, M., Subhan, F., Ahmad, N., Ali, G., Akbar, S., Fawad, K. and Sewell, Robert David Edmund 2017. Topical gabapentin gel alleviates allodynia and hyperalgesia in the chronic sciatic nerve constriction injury neuropathic pain model. European Journal of Pain 21 (4) , pp. 668-680. 10.1002/ejp.971

Shahid, Muhammad, Subhan, Fazal, Ahmad, Nisar and Sewell, Robert D. E. 2017. The flavonoid 6-methoxyflavone allays cisplatin-induced neuropathic allodynia and hypoalgesia. Biomedicine & Pharmacotherapy 95 , pp. 1725-1733. 10.1016/j.biopha.2017.09.108

Singh, Ravinder, Perks, William, Twohig, Jason, Kidd, Emma

, Broadley, Kenneth

, Farrow, S N, Williams, Anwen

, Taylor, Philip

and Wang, Edward

2017. Death receptor 3 regulates distinct pathological attributes of acute versus chronic murine allergic lung inflammation. Cellular Immunology 320 , pp. 62-70. 10.1016/j.cellimm.2017.09.005

Somasagara, R. R., Spencer, S. M., Tripathi, K., Clark, D. W., Mani, C., Madeira da Silva, L., Scalici, J., Kothayer, H., Westwell, A. D.

, Rocconi, R. P. and Palle, K. 2017. RAD6 promotes DNA repair and stem cell signaling in ovarian cancer and is a promising therapeutic target to prevent and treat acquired chemoresistance. Oncogene 36 , pp. 6680-6690. 10.1038/onc.2017.279

Spark, J M, Tawil, R, O'Brien, B, Sutherland-Plozza, Z, Charles, S and John, David

2017. What are the attributes of good pharmacy faculty (lecturers)? An international comparison of the views of pharmacy undergraduate students from universities in Australia and Wales, UK. Pharmacy Education 17 (1) , pp. 36-42.

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Taban, Ismail 2017. Design and synthesis of novel CYP24A1 inhibitors. PhD Thesis, Cardiff University.

Item availability restricted.

Taban, Ismail M., Zhu, Jing, DeLuca, Hector F. and Simons, Claire

2017. Analysis of the binding sites of vitamin D 1α-hydroxylase (CYP27B1) and vitamin D 24-hydroxylase (CYP24A1) for the design of selective CYP24A1 inhibitors: homology modelling, molecular dynamics simulations and identification of key binding requirements. Bioorganic & Medicinal Chemistry 25 (20) , pp. 5629-5636. 10.1016/j.bmc.2017.08.036

Taban, Ismail M., Zhu, Jinge, DeLuca, Hector F. and Simons, Claire

2017. Synthesis, molecular modelling and CYP24A1 inhibitory activity of novel of (E)-N-(2-(1H-imidazol-1-yl)-2-(phenylethyl)-3/4-styrylbenzamides. Bioorganic and Medicinal Chemistry 25 (15) , pp. 4076-4087. 10.1016/j.bmc.2017.05.055

Taban, Ismail, Elshihawy, Hosam A. E., Torun, Beyza, Zucchini, Benedetta, Williamson, Clare J., Altuwairigi, Dania, Ngu, Adeline S. T., McLean, Kirsty J., Levy, Colin W., Sood, Sakshi, Marino, Leonardo B., Munro, Andrew W., de Carvalho, Luiz Pedro S. and Simons, Claire

2017. Novel aryl substituted pyrazoles as small molecule inhibitors of cytochrome P450 CYP121A1: Synthesis and antimycobacterial evaluation. Journal of Medicinal Chemistry 60 (24) , pp. 10257-10267. 10.1021/acs.jmedchem.7b01562

Tamboli, Vibha 2017. Detection of prostate cancer biomarker using molecularly imprinted polymers. PhD Thesis, Cardiff University.

Item availability restricted.

Thomas, R.S., Alsaqati, Mouhamed, Bice, Justin, Hvoslef-Eide, M, Good, Mark

and Kidd, Emma

2017. Alterations in endocytic protein expression with increasing age in the transgenic APP695 V717I London mouse model of amyloid pathology - implications for Alzheimer's disease. NeuroReport 28 (15) , pp. 963-968. 10.1097/WNR.0000000000000861

Tochwin, Anna, El-Betany, Alaa

, Tai, Hongyun, Chan, Kai, Blackburn, Chester and Wang, Wenxin 2017. Thermoresponsive and reducible hyperbranched polymers synthesized by RAFT polymerisation. Polymers 9 (9) , 443. 10.3390/polym9090443

Tuncay, Erkan, Bitirim, Verda C., Durak, Aysegul, Carrat, Gaelle R.J., Taylor, Kathryn

, Rutter, Guy A. and Turan, Belma 2017. Hyperglycemia-induced changes in ZIP7 and ZnT7 expression cause Zn2+ release from the sarco(endo)plasmic reticulum and mediate ER-stress in the heart. Diabetes 66 (5) , pp. 1346-1358. 10.2337/db16-1099

Turner, Dawn L., Ford, William R.

, Kidd, Emma J.

, Broadley, Kenneth J.

and Powell, Colin 2017. Effects of nebulised magnesium sulphate on inflammation and function of the guinea-pig airway. European Journal of Pharmacology 801 , pp. 79-85. 10.1016/j.ejphar.2017.03.004

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Wong, Pei Nee 2017. A mixed methods approach for assessing student and staff perceptions and experiences of a new collaborative transnational pharmacy programme. PhD Thesis, Cardiff University.

Item availability restricted.

Wymant, Jennifer, Moody, P., Sayers, Edward

and Jones, Arwyn Tomos

2017. Poster 433: Receptor-antibody clustering induced endocytosis of HER2 has therapeutic potential in breast cancer. Presented at: EACR-AACR-SIC Special Conference 2017: The Challenges of Optimising Immuno and Targeted Therapies From Cancer Biology to the Clinic, Florence, Italy, 24-27 June 2017.

Y

Yemm, Rowan

, Jones, Christabel and Mitoko, Tryphosa 2017. Displaying medication costs on dispensing labels as a strategy to reduce wastage: views of the Welsh general public. Integrated Pharmacy Research and Practice 6 , pp. 173-180. 10.2147/IPRP.S145567

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Zhao, Xin, Coulman, Sion A.

, Hanna, Stephanie J., Wong, F. Susan

, Dayan, Colin M.

and Birchall, James C.

2017. Formulation of hydrophobic peptides for skin delivery via coated microneedles. Journal of Controlled Release 265 , pp. 2-13. 10.1016/j.jconrel.2017.03.015

Zheng, Chen 2017. The use of excipients to stabilise pressurised metered dose inhalers. PhD Thesis, Cardiff University.

Item availability restricted.

Ziedan, Noha I, Hamdy, Rania, Cavaliere, Alessandra, Kourti, Malamati, Prencipe, Filippo, Brancale, Andrea

, Jones, Arwyn T

and Westwell, Andrew

2017. Virtual screening, SAR and discovery of 5-(indole-3-yl)-2-[(2-nitrophenyl)amino] [1,3,4]-oxadiazole as a novel Bcl-2 inhibitor. Chemical Biology and Drug Design 10.1111/cbdd.12936

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